The metabolism of some substituted benzofuran β-adrenergic blocking agents
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چکیده
منابع مشابه
Femoral vascular effects of some beta receptor adrenergic blocking agents.
Beta receptor adrenergic blocking agents produce a fall of systemic arterial blood pressure which has been attributed to interference with the function of sympathetic nerves to the heart (1). While pronethalol and propranolol are known to have a peripheral vasodilator component of action which contributes to their hypo tensive effect (2, 3), it has not been determined if the more recently synth...
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Cardiac dysfunction in heart failure is widely recognized as a progressive process, regardless of the clinical signs and symptoms. An increase in cardiac sympathetic drive is one of the earliest neurohormonal responses occurring in patients with heart failure and may be one of the major causes of the progressive remodeling leading to the decline in myocardial function, and responsible for the p...
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Performance anxiety consists qf several symptoms experienced in the context qf public performance and is classified in DSM-III-R under social phobia. Performance anxiety must be distinguished from panic disorder, generalized social phobia, and generalized anxiety disorder. Petformance anxiety symptoms can be detrimental to both petformer and performance. These symptoms can be controlled by the ...
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In this investigation, the synthesis of 2-substituted pyrimidines by the reaction of benzofuranchalcones (3a-d) with urea, thiourea and guanidine hydrochloride was reported. The structuresof title compounds (4a-d), (5a-d) and (6a-d) were established on the basis of analyticaland spectral data. The synthesized compounds were screened for antimicrobial activityand molecular docking studies. Some ...
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ژورنال
عنوان ژورنال: Biochemical Journal
سال: 1969
ISSN: 0306-3283
DOI: 10.1042/bj1150060pa